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Bepridil


Bepridil
Systematic (IUPAC) name
(±)-(beta)-[(2-Methylpropoxy)methyl]-N-phenyl- N -(phenyl- methyl)-1-pyrrolidineethanamine
Identifiers
CAS number	64706-54-3
ATC code	C08EA02
PubChem	2351
DrugBank	APRD00727
Chemical data
Formula	C₂₄H₃₄N₂O
Mol. mass	421.02 g/mol
Pharmacokinetic data
Bioavailability	Well absorbed
Protein binding	99%
Metabolism	Hepatic, CYP3A4-mediated
Half life	42 hours
Excretion	Renal
Therapeutic considerations
Pregnancy cat.	C(US)
Legal status
Routes	Oral

Bepridil (trade name Vascor) is a calcium channel blocker once used to treat angina. It is no longer sold in the United States.

v • d • e Calcium channel blockers (C08)
Dihydropyridines	Amlodipine • Felodipine • Isradipine • Lacidipine • Lercanidipine • Nicardipine • Nifedipine • Nimodipine • Nisoldipine • Nitrendipine
Phenylalkylamines	Verapamil
Benzothiazepines	Diltiazem