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Ipsapirone


Ipsapirone
Systematic (IUPAC) name
9,9-Dioxo-8-[4-(4-pyrimidin-2-ylpiperazin-1-yl)butyl]- 9λ⁶-thia-8-azabicyclo[4.3.0]nona-1,3,5-trien-7-one
Identifiers
CAS number	95847-70-4
ATC code	?
PubChem	56971
Chemical data
Formula	C₁₉H₂₃N₅O₃S
Mol. mass	401.484 g/mol
Pharmacokinetic data
Bioavailability	?
Metabolism	?
Half life	?
Excretion	?
Therapeutic considerations
Pregnancy cat.	?
Legal status
Routes	?

Ipsapirone is an azapirone and partial 5-HT1A agonist that has anxiolytic effects.

References

Fanelli R, Schuurman T, Glaser T, Traber J (1990). "Ipsapirone: a novel anxiolytic and selective 5-HT1A receptor ligand.". Prog Clin Biol Res 361: 461–7. PMID 1981264.