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Carteolol


Carteolol
Systematic (IUPAC) name
5-[2-hydroxy-3- (tert-butylamino) propoxy]- 3,4-dihydro-1H-quinolin-2-one
Identifiers
CAS number	51781-06-7
ATC code	C07AA15 S01ED05
PubChem	2583
DrugBank	APRD00195
Chemical data
Formula	C₁₆H₂₄N₂O₃
Mol. mass	292.373 g/mol
Pharmacokinetic data
Bioavailability	85%
Metabolism	hepatic, active with 8-hyrdocarteolol
Half life	6-8 hours
Excretion	Renal (50-70%)
Therapeutic considerations
Pregnancy cat.	C(US)
Legal status
Routes	oral

Carteolol is a beta blocking agent

v • d • e Ophthalmologicals: antiglaucoma preparations and miotics (S01E)
Sympathomimetics	Apraclonidine • Brimonidine • Clonidine • Dipivefrine • Epinephrine
Parasympathomimetics	Aceclidine • Acetylcholine • Carbachol • Demecarium • Echothiophate • Stigmine (Fluostigmine, Neostigmine, Physostigmine) • Paraoxon • Pilocarpine
Carbonic anhydrase inhibitors	Acetazolamide • Brinzolamide • Diclofenamide • Dorzolamide • Methazolamide
Beta blocking agents	Befunolol • Betaxolol • Carteolol • Levobunolol • Metipranolol • Timolol
Prostaglandin analogues	Bimatoprost • Latanoprost • Travoprost • Unoprostone
Other agents	Dapiprazole • Guanethidine